⚗️ Drug Safety Research

Drug Interactions Guide — 21 Medications with Severity Ratings

FDA prescribing information sourced. Every interaction rated dangerous, serious, or moderate — so you know what to ask your doctor.

37
Dangerous interactions documented
48
Serious interactions documented
19
Moderate interactions documented
21
Drugs covered
What Are Drug Interactions?

A drug interaction occurs when one substance changes the effect of another drug in the body — either increasing its potency (sometimes to toxic levels), decreasing its effectiveness, or producing entirely new effects. Interactions can occur between two prescription drugs, between a drug and an over-the-counter medication, or between a drug and food, alcohol, or a supplement.

The consequences range from minor inconveniences to life-threatening emergencies. Some interactions — like opioids combined with benzodiazepines — have killed thousands of people. Others require only modest monitoring adjustments. Understanding the severity of a specific interaction is the difference between a conversation with your doctor and an emergency room visit.

⚠️ Most interactions are preventable The leading cause of preventable drug interaction harm is patients receiving prescriptions from multiple prescribers who don't share records, or failing to disclose OTC drugs, alcohol, and supplements. A complete medication list — shared with every provider and pharmacist — eliminates the majority of interaction risk.

PillScope's interaction data is sourced from FDA-approved prescribing information (the "package insert") for each medication. Severity ratings reflect FDA classification, clinical severity in published case reports, and whether the interaction appears in the contraindication versus warning-and-precaution sections of the label.

How Drug Interactions Cause Harm
⚗️

Metabolic (CYP Enzyme) Interactions

Most drug metabolism happens in the liver via CYP450 enzymes. When one drug blocks these enzymes, another drug accumulates to toxic levels. Warfarin, fentanyl, statins, and benzodiazepines are all processed by CYP enzymes — a common source of dangerous interactions.

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Additive CNS Depression

Two drugs that each slow the central nervous system — opioids, benzodiazepines, alcohol, sleep aids, muscle relaxants — stack synergistically. The combination can stop breathing entirely at doses that would individually be survivable. This is the mechanism behind most prescription overdose deaths.

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QT Interval Prolongation

Some drugs extend the heart's electrical recovery time (QT interval). When multiple QT-prolonging drugs combine — methadone, antipsychotics, fluoroquinolones, certain antidepressants — the risk of fatal ventricular arrhythmia (torsades de pointes) escalates sharply.

21 Drugs Sorted by Interaction Severity
Dangerous — Life-threatening; may be contraindicated
Serious — Significant harm; requires monitoring or dose adjustment
Moderate — Notable; awareness and monitoring advised
1
🧘 Xanax alprazolam Benzodiazepine
4 dangerous1 serious5 interactions documented
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2
💊 Fentanyl fentanyl Opioid
4 dangerous1 serious5 interactions documented
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3
💊 Methadone methadone Opioid
3 dangerous2 serious5 interactions documented
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4
💊 OxyContin oxycodone Opioid
3 dangerous2 serious5 interactions documented
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5
🧘 Klonopin clonazepam Benzodiazepine
3 dangerous1 serious1 moderate5 interactions documented
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6
🫀 Lipitor atorvastatin Statin
3 dangerous1 serious1 moderate5 interactions documented
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7
🩸 Warfarin warfarin Anticoagulant
2 dangerous2 serious1 moderate5 interactions documented
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8
💊 Tramadol tramadol Opioid
2 dangerous3 serious5 interactions documented
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9
🧘 Valium diazepam Benzodiazepine
2 dangerous2 serious1 moderate5 interactions documented
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10
🧘 Ativan lorazepam Benzodiazepine
2 dangerous2 serious1 moderate5 interactions documented
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11
🧬 Methotrexate methotrexate DMARD
2 dangerous3 serious5 interactions documented
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12
🦠 Levaquin levofloxacin Fluoroquinolone
1 dangerous2 serious2 moderate5 interactions documented
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13
🦠 Avelox moxifloxacin Fluoroquinolone
1 dangerous2 serious2 moderate5 interactions documented
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14
🧠 Seroquel quetiapine Antipsychotic
1 dangerous2 serious2 moderate5 interactions documented
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15
🧠 Zyprexa olanzapine Antipsychotic
1 dangerous3 serious1 moderate5 interactions documented
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16
Ritalin methylphenidate Stimulant
1 dangerous2 serious2 moderate5 interactions documented
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17
🦠 Cipro ciprofloxacin Fluoroquinolone
1 dangerous3 serious1 moderate5 interactions documented
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18
🔥 Celebrex celecoxib NSAID
1 dangerous4 serious5 interactions documented
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19
🧠 Abilify aripiprazole Antipsychotic
3 serious2 moderate5 interactions documented
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20
💊 Accutane isotretinoin Retinoid
3 serious1 moderate4 interactions documented
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21
⚠️ Vioxx rofecoxib NSAID (withdrawn)
4 serious1 moderate5 interactions documented
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Drug Interactions FAQ
Medical Disclaimer: PillScope provides educational information only. This page is not medical advice. Do not stop, start, or change any medication based on this information without consulting your doctor or pharmacist. Interaction data is sourced from FDA prescribing information and may not reflect all possible interactions for your specific situation.